ClinicalTrials.Veeva

Menu

Linking Altered Central Pain Processing and Genetic Polymorphism to Drug Efficacy in Chronic Low Back Pain (Predictio)

I

Insel Gruppe AG, University Hospital Bern

Status and phase

Completed
Phase 3

Conditions

Low Back Pain

Treatments

Drug: Tolterodine
Drug: Imipramine
Drug: Oxycodone 15mg
Drug: Clobazam

Study type

Interventional

Funder types

Other

Identifiers

NCT01179828
KEK 213/09
grant: SPUM no. 33CM30_124117

Details and patient eligibility

About

Drug therapy in patients with chronic low back pain is a major challenge for physicians. One of the problems is the lacking knowledge in prediction of drug efficacy in a chosen patient. Usually one of the classes of pain medication is given to patients with a similar clinical picture, although different pain mechanisms may be responsible for this clinical picture.

Another reason for variable drug efficacy are genetic polymorphisms, this may be the reason why an unique drug produces different responses (from a lacking analgesic effect up to excessive effect or side-effects.

Quantitative sensory testing is a method that documents alterations in the pain perception system. Linking genetic polymorphisms to quantitative sensory testing may give us a tool for anticipation of drug efficacy.

Full description

Background

Drug therapy is an essential part of pain treatment. However, only a minor part of pain patients benefits from the available treatments or is able to tolerate the drugs. One important limitation of drug therapy is lack of instruments to predict their effect. Indeed, in clinical practice "classes" of drugs (e.g. antidepressants) are given to "classes" of patients (e.g. neuropathic pain patients). However, within those classes of patients very different pain mechanisms are likely to underlie the pain condition in different patients. If drugs affect part of these mechanisms, they will not work in all patients. Another reason for variability in drug responses is genetic variation leading to a spectrum of different responses to analgesics, from lack of efficacy to exaggerated responses, up to intolerable adverse effects.

Quantitative sensory testing comprises methods that document alterations and reorganization of the nociceptive system. Measuring an abnormal result in a chronic pain patient may provide us with the information that the underlying pain pathways somehow must be altered. An essential question is whether this information can be linked to drug efficacy in a mechanism-based treatment approach. A further important question is whether assessing genetic polymorphisms can explain different drug effects and hence help selecting the appropriate therapeutic strategy for individual patients.

Objective

We will test the hypothesis that there is a correlation between disturbances in specific pain mechanisms as assessed by quantitative sensory tests and analgesic efficacy after single-dose drug administration in patients with chronic low back pain. Genetic factors affecting drug metabolism and pain sensitivity will be analyzed as additional explanatory variables for drug efficacy.

Methods

Quantitative sensory testing: Heat pain threshold and tolerance, Ice water testing with central modulation of nociceptive input (DNIC), electrical pain detection and temporal summation (skin probe), pressure algometry with pain detection and threshold Drugs investigated: Imipramine, Oxycodone, Clobazam Blood samples: pharmacogenetics: Cytochrome variants CYP2D6, CYP2C19, CYP3A4, COMT haplotypes, CGH-1 variants, A118G of mu opioid receptor gene variants pharmacokinetics: kinetics of imipramine and desipramine

Enrollment

150 patients

Sex

All

Ages

18 to 80 years old

Volunteers

No Healthy Volunteers

Inclusion and exclusion criteria

Inclusion Criteria:

  • Low back pain with NRS>2
  • Chronic low back pain since more than 6 months

Exclusion Criteria

  • pregnancy
  • use of pain medication other than paracetamol and ibuprofen in the last 7 days
  • suspicion of radicular pain
  • suspicion of intervertebral disk herniation
  • foraminal intervertebral stenosis
  • suspicion of polyneuropathy
  • diabetes
  • parkinson disease
  • alzheimer disease
  • glaucoma
  • prostata hyperplasia or voiding problems
  • known heart rhythm problems
  • heart insufficiency NYHA 3-4
  • Systemic inflammatory disease
  • Ongoing oncologic disease
  • drug or alcohol abuse
  • Significant depressive disease (BDI-FS>9)

Trial design

Primary purpose

Basic Science

Allocation

Randomized

Interventional model

Crossover Assignment

Masking

Triple Blind

150 participants in 4 patient groups, including a placebo group

1
Active Comparator group
Description:
Oxycodone 15mg
Treatment:
Drug: Oxycodone 15mg
2
Active Comparator group
Description:
Clobazam 20mg
Treatment:
Drug: Clobazam
3
Active Comparator group
Description:
Imipramine 75mg
Treatment:
Drug: Imipramine
4
Placebo Comparator group
Description:
Tolterodine 1mg
Treatment:
Drug: Tolterodine

Trial contacts and locations

1

Loading...

Data sourced from clinicaltrials.gov

Clinical trials

Find clinical trialsTrials by location
© Copyright 2026 Veeva Systems